Clobazam
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| TripSit | Pharmacology | DrugCentral | DailyMed | ||
|---|---|---|---|---|---|
| Classification | |||||
| Class / category | — | — | — | ||
| Also known as | frisium | — | — | — | |
| Safety | |||||
| Dose · Oral | |||||
| Light | 5–10 mg | — | — | — | |
| Common | 10–15 mg | — | — | — | |
| Heavy | 15 mg+ | — | — | — | |
| Duration | |||||
| Onset | 20–40 minutes | — | — | — | |
| Total | 6–12 hours | — | — | — | |
| After-effects | 1–12 hours | — | — | — | |
| Pharmacology | |||||
| Receptor activity | — | — | GABRA1 | — | |
| Half-life | — | The estimated mean elimination half-lives (t½) of clobazam and N-desmethylclobazam were 36-42 hours and 71-82 hours, respectively. The mean elimination half-life of clobazam is approximately 36-42 hours and the mean elimination half-life of N-desmethylclobazam is approximately 71-82 hours. | — | — | |
| Protein binding | — | The in vitro plasma protein binding of clobazam and N-desmethylclobazam is approximately 80-90% and 70%, respectively. | — | — | |
TripSit summary
A long acting benzodiazepine which focuses primarily on anxiolytic and anticonvulsant properties. It is used medically to treat epilepsy, and this along with its relatively many negative side-effects and contraindications in comparison with other benzodiazepines means it isn't frequently used recreationally.
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.