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Flunitrazepam

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🧬 Receptor activity

TargetActionAffinitySource
Gamma-aminobutyric acid receptor subunit alpha-1 (GABRA1)Allosteric modulator8.28 KiDRUGCENTRAL
Gamma-aminobutyric acid receptor subunit alpha-2 (GABRA2)Allosteric modulator8.28 KiDRUGCENTRAL
Gamma-aminobutyric acid receptor subunit alpha-3 (GABRA3)Allosteric modulator7.8 KiDRUGCENTRAL
Gamma-aminobutyric acid receptor subunit alpha-5 (GABRA5)Allosteric modulator8.26 KiDRUGCENTRAL
GABA A receptor alpha-3/beta-2/gamma-2 (GABRG2)8.824 KiDRUGCENTRAL
GABA A receptor alpha-3/beta-2/gamma-3 (GABRA3)7.5 KiDRUGCENTRAL
GABA A receptor alpha-5/beta-2/gamma-2 (GABRG2)9 KiDRUGCENTRAL
GABA A receptor alpha-5/beta-2/gamma-3 (GABRA5)8.42 KiDRUGCENTRAL
GABA A receptor alpha-5/beta-3/gamma-3 (GABRB3)8.42 KiDRUGCENTRAL
GABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1)8.699 KiDRUGCENTRAL
GABA-A receptor alpha-1/beta-2/gamma-3 (GABRA1)7.457 KiDRUGCENTRAL
GABA-A receptor alpha-1/beta-3/gamma-2 (GABRA1)8.47 KiDRUGCENTRAL
GABA-A receptor alpha-2/beta-3/gamma-2 (GABRG2)8.699 KiDRUGCENTRAL
GABA-A receptor alpha-3/beta-3/gamma-2 (GABRG2)8.347 KiDRUGCENTRAL
GABA-A receptor alpha-5/beta-3/gamma-2 (GABRG2)8.84 KiDRUGCENTRAL
GABA-A receptor; anion channel (Gabrp)8.82 IC50DRUGCENTRAL
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Source: DrugCentral — Flunitrazepam ↗

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