Medazepam
Discover related
3 sources
Collated from TripSit, Pharmacology, DrugCentral. Where sources differ (e.g. dosing), Compare shows them side by side.
Also known as nobrium, azepamid, rudotel, raporan, mezapam, talisTS
Benzodiazepine derivative that has all of the classic benzodiazepine effects. Is a long-acting benzodiazepine drug (Half life of 36-200 hours) Is rarely prescribed in most countries. Is also a prodrug for Diazepam. Think of it as Desoxy-Diazepam if you'd like to.TS
Oral
Route dataTripSit
| Threshold | Light | Common | Strong | Heavy |
|---|---|---|---|---|
| — | 5–10 mg | 10–20 mg | 20–40 mg | —+ |
040 mg
LightCommonStrongHeavy
| Onset | 30–120 minutes |
|---|---|
| Total | 8–16 hours |
| After-effects | 1–172 hours |
OnsetCome-upPeakOffset
🧬 Receptor activityPHDC
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA-A receptor; anion channel | — | Ki 528 nM | CHEMBL | TargetGABA-A receptor; anion channel Action— AffinityKi 528 nM SourceCHEMBL |
| GABA-A receptor; anion channel (Gabrp) | — | 6.28 Ki | DRUGCENTRAL | TargetGABA-A receptor; anion channel (Gabrp) Action— Affinity6.28 Ki SourceDRUGCENTRAL |
Plan when to take Medazepam — see where onset, peak and comedown land on the clock
Plan a dose of Medazepam
Loading the fact-sheet…
Logging a dose needs somewhere to keep it. Start a free session — no signup; it and everything in it expire in 7 days.
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.