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Nordazepam

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3 sources

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Collated from TripSit, Pharmacology, DrugCentral. Where sources differ (e.g. dosing), Compare shows them side by side.

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BenzodiazepineHabit-formingDepressantTS

Also known as nordaz, nordiazepam, desmethyldiazepamTS

Has all the normal benzodiazepine effects. Such as being an anti-convulsant, muscle relaxant, sedative effects, and anxiolytic. Active metabolite of Diazepam, Chlordiazepoxide, Clorazepate, among many others, which is where most of its effects come from. Has one of the longest lasting half-lifes in the class.TS

Oral

Route dataTripSit

Dose
WeakerStronger
ThresholdLightCommonStrongHeavy
—2.5–5 mg5–15 mg15–30 mg—+
030 mg
LightCommonStrongHeavy
Duration
ShorterLonger
Onset45–120 minutes
Total10–20 hours
After-effects1–120 hours
OnsetCome-upPeakOffset

🧬 Receptor activityPHDC

TargetActionAffinitySource
GABA-A receptor; anion channel—Ki 73000 nMCHEMBL
GABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1)—6.284 IC50DRUGCENTRAL
GABA-A receptor; anion channel (Gabre)—4.14 KiDRUGCENTRAL
Gamma-aminobutyric acid receptor subunit rho-2 (GABRR2)——DRUGCENTRAL
Gamma-aminobutyric acid type B receptor subunit 2 (GABBR2)—8.027 IC50DRUGCENTRAL
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Pharmacokinetics

MetabolismPH

Nordiazepam has known human metabolites that include Oxazepam.
Nordiazepam is a known human metabolite of diazepam.

Plan when to take Nordazepam — see where onset, peak and comedown land on the clock

Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.