Zolpidem
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) | Positive allosteric modulator | 6.164 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity6.164 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) | Positive allosteric modulator | 6.703 EC50 | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) ActionPositive allosteric modulator Affinity6.703 EC50 SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-3/gamma-2 (GABRA1) | Positive allosteric modulator | 7.574 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-3/gamma-2 (GABRA1) ActionPositive allosteric modulator Affinity7.574 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-2/beta-3/gamma-2 (GABRG2) | Positive allosteric modulator | 6.807 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-2/beta-3/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity6.807 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-3/beta-3/gamma-2 (GABRG2) | Positive allosteric modulator | 6.417 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-3/beta-3/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity6.417 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-1 (GABRA1) | Allosteric modulator | 7.68 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-1 (GABRA1) ActionAllosteric modulator Affinity7.68 Ki SourceDRUGCENTRAL |
| CAAX prenyl protease 2 (RCE1) | — | 4.77 AC50 | DRUGCENTRAL | TargetCAAX prenyl protease 2 (RCE1) Action— Affinity4.77 AC50 SourceDRUGCENTRAL |
| GABA A receptor alpha-2/beta-2/gamma-2 (Gabrg2) | — | 6.81 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-2/beta-2/gamma-2 (Gabrg2) Action— Affinity6.81 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-3/beta-2/gamma-2 (Gabrg2) | — | 6.42 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-2 (Gabrg2) Action— Affinity6.42 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-6/beta-2/gamma-2 (Gabrg2) | — | 6.01 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-6/beta-2/gamma-2 (Gabrg2) Action— Affinity6.01 Ki SourceDRUGCENTRAL |
| GABA-A receptor; alpha-1/beta-2/gamma-2 (Gabrg2) | — | 7.72 Ki | DRUGCENTRAL | TargetGABA-A receptor; alpha-1/beta-2/gamma-2 (Gabrg2) Action— Affinity7.72 Ki SourceDRUGCENTRAL |
| GABA-A receptor; anion channel (Gabrp) | — | 7.6 Ki | DRUGCENTRAL | TargetGABA-A receptor; anion channel (Gabrp) Action— Affinity7.6 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-1 (Gabra1) | — | 7.3 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-1 (Gabra1) Action— Affinity7.3 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-2 (GABRA2) | — | 6.39 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-2 (GABRA2) Action— Affinity6.39 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-3 (GABRA3) | — | 6.01 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-3 (GABRA3) Action— Affinity6.01 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-5 (Gabra5) | — | 7.46 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-5 (Gabra5) Action— Affinity7.46 Ki SourceDRUGCENTRAL |
| Multidrug resistance protein 1 (ABCB1) | — | 3.703 Km | DRUGCENTRAL | TargetMultidrug resistance protein 1 (ABCB1) Action— Affinity3.703 Km SourceDRUGCENTRAL |
| Translocator protein (Tspo) | — | 5.33 IC50 | DRUGCENTRAL | TargetTranslocator protein (Tspo) Action— Affinity5.33 IC50 SourceDRUGCENTRAL |
External links
PubChem 5732 ↗CAS 82626-48-0 ↗KEGG C07219 ↗ChEBI CHEBI:10125 ↗ChEMBL CHEMBL911 ↗KEGG D08690 ↗DrugBank DB00425 ↗ChemSpider ↗ChEBI/ChEMBL ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗Guide to Pharmacology ↗NIH ↗NIH ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗CAS 103188-50-7 ↗CAS 43200-81-3 ↗CAS 82628-28-2 ↗CAS 959605-90-4 ↗CAS 99294-93-6 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Zolpidem ↗
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.