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🧬 Receptor activity

TargetActionAffinitySource
Adenosine receptor A1 (ADORA1)Antagonist4.97 KiDRUGCENTRAL
Adenosine receptor A2a (ADORA2A)Antagonist5.61 KiDRUGCENTRAL
Adenosine receptor A2b (ADORA2B)Antagonist4.77 KiDRUGCENTRAL
Adenosine receptor A3 (ADORA3)Antagonist4.33 KiDRUGCENTRAL
Acetylcholinesterase (ACHE)5.14 IC50DRUGCENTRAL
Adenosine A2 receptor (Adora2b)4.57 KiDRUGCENTRAL
Adenosine A2a receptor (ADORA2A)4.1 KiDRUGCENTRAL
Adenosine receptor (Adora1)4.22 KiDRUGCENTRAL
Adenosine receptor A1 (Adora1)4.77 KiDRUGCENTRAL
Adenosine receptor A2a (Adora2a)5.03 KiDRUGCENTRAL
Glycogen phosphorylase, muscle form (PYGM)4.13 IC50DRUGCENTRAL
Guanine deaminase (GDA)4.99 KiDRUGCENTRAL
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform (PIK3CD)4.12 IC50DRUGCENTRAL
Potassium voltage-gated channel subfamily H member 2 (KCNH2)5.31 IC50DRUGCENTRAL
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Source: DrugCentral — Caffeine ↗

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