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Cinolazepam

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🔗 MergedCompareTripSitPharmacology

Collated from TripSit, Pharmacology. Where sources differ (e.g. dosing), Compare shows them side by side.

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DepressantHabit-formingTS

Also known as gerodermTS

A benzodiazepine derivative drug with anxiolytic effects but mainly hypnotic effects. It is extremely effective for sleep aid but has mild euphoria compared to other benzosTS

Oral

Route dataTripSit

Dose
WeakerStronger
ThresholdLightCommonStrongHeavy
—10–30 mg30–60 mg60–120 mg—+
0120 mg
LightCommonStrongHeavy
Duration
ShorterLonger
Onset30–90 minutes
Total8–12 hours
After-effects12–20 hours
OnsetCome-upPeakOffset

Mechanism of actionPH

Cinolazepam binds to central benzodiazepine receptors which interact allosterically with GABA receptors. This potentiates the effects of the inhibitory neurotransmitter GABA, increasing the inhibition of the ascending reticular activating system and blocking the cortical and limbic arousal that occurs following stimulation of the reticular pathways.

PharmacodynamicsPH

Cinolazepam is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. It is not approved in Canada or America.

Pharmacokinetics

Half-lifePH

9 hours

AbsorptionPH

Bioavailability following oral administration is 90-100%.

MetabolismPH

Hepatic.
Hepatic.
Half Life: 9 hours

Plan when to take Cinolazepam — see where onset, peak and comedown land on the clock

Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.