Cyclobenzaprine
Discover related
4 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| 5-hydroxytryptamine receptor 2A (HTR2A) | Antagonist | 7.541 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 2A (HTR2A) ActionAntagonist Affinity7.541 Ki SourceDRUGCENTRAL |
| 5-hydroxytryptamine receptor 2C (HTR2C) | Antagonist | 7.244 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 2C (HTR2C) ActionAntagonist Affinity7.244 Ki SourceDRUGCENTRAL |
| 5-hydroxytryptamine receptor 2B (HTR2B) | — | 6.812 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 2B (HTR2B) Action— Affinity6.812 Ki SourceDRUGCENTRAL |
| 5-hydroxytryptamine receptor 6 (HTR6) | — | 6.839 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 6 (HTR6) Action— Affinity6.839 Ki SourceDRUGCENTRAL |
| 5-hydroxytryptamine receptor 7 (HTR7) | — | 6.821 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 7 (HTR7) Action— Affinity6.821 Ki SourceDRUGCENTRAL |
| Aldehyde oxidase (AOX1) | — | 5.509 IC50 | DRUGCENTRAL | TargetAldehyde oxidase (AOX1) Action— Affinity5.509 IC50 SourceDRUGCENTRAL |
| Histamine H1 receptor (HRH1) | — | 8.829 Ki | DRUGCENTRAL | TargetHistamine H1 receptor (HRH1) Action— Affinity8.829 Ki SourceDRUGCENTRAL |
| Multidrug resistance protein 1 (ABCB1) | — | 4.728 IC50 | DRUGCENTRAL | TargetMultidrug resistance protein 1 (ABCB1) Action— Affinity4.728 IC50 SourceDRUGCENTRAL |
| Muscarinic acetylcholine receptor M1 (CHRM1) | — | 6.95 IC50 | DRUGCENTRAL | TargetMuscarinic acetylcholine receptor M1 (CHRM1) Action— Affinity6.95 IC50 SourceDRUGCENTRAL |
| Muscarinic acetylcholine receptor M2 (CHRM2) | — | 7.222 Ki | DRUGCENTRAL | TargetMuscarinic acetylcholine receptor M2 (CHRM2) Action— Affinity7.222 Ki SourceDRUGCENTRAL |
| Muscarinic acetylcholine receptor M3 (CHRM3) | — | 8.222 Ki | DRUGCENTRAL | TargetMuscarinic acetylcholine receptor M3 (CHRM3) Action— Affinity8.222 Ki SourceDRUGCENTRAL |
| Proto-oncogene tyrosine-protein kinase receptor Ret (RET) | — | 6.52 IC50 | DRUGCENTRAL | TargetProto-oncogene tyrosine-protein kinase receptor Ret (RET) Action— Affinity6.52 IC50 SourceDRUGCENTRAL |
| Sodium-dependent noradrenaline transporter (SLC6A2) | — | 7.444 Ki | DRUGCENTRAL | TargetSodium-dependent noradrenaline transporter (SLC6A2) Action— Affinity7.444 Ki SourceDRUGCENTRAL |
| Sodium-dependent serotonin transporter (SLC6A4) | — | 6.967 Ki | DRUGCENTRAL | TargetSodium-dependent serotonin transporter (SLC6A4) Action— Affinity6.967 Ki SourceDRUGCENTRAL |
External links
PubChem 2895 ↗CAS 303-53-7 ↗KEGG C06931 ↗ChEBI CHEBI:3996 ↗ChEMBL CHEMBL669 ↗KEGG D07758 ↗DrugBank DB00924 ↗NIH ↗NIH ↗NIH ↗ChemSpider ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗CAS 6202-23-9 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Cyclobenzaprine ↗
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