Eszopiclone
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| GABA A receptor alpha-3/beta-2/gamma-3 (GABRA3) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-3 (GABRA3) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| GABA A receptor alpha-5/beta-2/gamma-2 (GABRG2) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA A receptor alpha-5/beta-2/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| GABA A receptor alpha-5/beta-2/gamma-3 (GABRA5) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA A receptor alpha-5/beta-2/gamma-3 (GABRA5) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-2/gamma-3 (GABRA1) | Positive allosteric modulator | — | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-2/gamma-3 (GABRA1) ActionPositive allosteric modulator Affinity— SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-2 (GABRA2) | Positive allosteric modulator | 6.94 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-2 (GABRA2) ActionPositive allosteric modulator Affinity6.94 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-4 (GABRA4) | Positive allosteric modulator | 6.99 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-4 (GABRA4) ActionPositive allosteric modulator Affinity6.99 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-1 (GABRA1) | — | 7.3 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-1 (GABRA1) Action— Affinity7.3 Ki SourceDRUGCENTRAL |
| Gamma-aminobutyric acid receptor subunit alpha-3 (GABRA3) | — | 6.79 Ki | DRUGCENTRAL | TargetGamma-aminobutyric acid receptor subunit alpha-3 (GABRA3) Action— Affinity6.79 Ki SourceDRUGCENTRAL |
External links
PubChem 969472 ↗CAS 138729-47-2 ↗ChEBI CHEBI:53760 ↗ChEMBL CHEMBL1522 ↗KEGG D02624 ↗DrugBank DB00402 ↗ChemSpider ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗NIH ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗CAS 1140433-81-3 ↗CAS 138680-08-7 ↗CAS 43200-80-2 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Eszopiclone ↗
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