Midazolam
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) | Positive allosteric modulator | 8.444 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity8.444 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-3/beta-2/gamma-3 (GABRA3) | Positive allosteric modulator | 7.613 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-3/beta-2/gamma-3 (GABRA3) ActionPositive allosteric modulator Affinity7.613 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-5/beta-2/gamma-2 (GABRG2) | Positive allosteric modulator | 9.125 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-5/beta-2/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity9.125 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-5/beta-2/gamma-3 (GABRA5) | Positive allosteric modulator | 8.26 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-5/beta-2/gamma-3 (GABRA5) ActionPositive allosteric modulator Affinity8.26 Ki SourceDRUGCENTRAL |
| GABA A receptor alpha-5/beta-3/gamma-3 (GABRB3) | Positive allosteric modulator | 8.26 Ki | DRUGCENTRAL | TargetGABA A receptor alpha-5/beta-3/gamma-3 (GABRB3) ActionPositive allosteric modulator Affinity8.26 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) | Positive allosteric modulator | 8.745 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-2/gamma-2 (GABRA1) ActionPositive allosteric modulator Affinity8.745 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-1/beta-2/gamma-3 (GABRA1) | Positive allosteric modulator | 7.75 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-1/beta-2/gamma-3 (GABRA1) ActionPositive allosteric modulator Affinity7.75 Ki SourceDRUGCENTRAL |
| GABA-A receptor alpha-5/beta-3/gamma-2 (GABRG2) | Positive allosteric modulator | 9.125 Ki | DRUGCENTRAL | TargetGABA-A receptor alpha-5/beta-3/gamma-2 (GABRG2) ActionPositive allosteric modulator Affinity9.125 Ki SourceDRUGCENTRAL |
| Thyrotropin-releasing hormone receptor (Trhr) | Antagonist | 5.49 Ki | DRUGCENTRAL | TargetThyrotropin-releasing hormone receptor (Trhr) ActionAntagonist Affinity5.49 Ki SourceDRUGCENTRAL |
| Cytochrome P450 3A4 (CYP3A4) | — | 6 Km | DRUGCENTRAL | TargetCytochrome P450 3A4 (CYP3A4) Action— Affinity6 Km SourceDRUGCENTRAL |
| GABA-A receptor; anion channel (Gabrp) | — | 8.7 Ki | DRUGCENTRAL | TargetGABA-A receptor; anion channel (Gabrp) Action— Affinity8.7 Ki SourceDRUGCENTRAL |
| Multidrug resistance protein 1 (ABCB1) | — | 4.353 Km | DRUGCENTRAL | TargetMultidrug resistance protein 1 (ABCB1) Action— Affinity4.353 Km SourceDRUGCENTRAL |
| Translocator protein (Tspo) | — | 8.7 Ki | DRUGCENTRAL | TargetTranslocator protein (Tspo) Action— Affinity8.7 Ki SourceDRUGCENTRAL |
External links
PubChem 4192 ↗CAS 59467-70-8 ↗KEGG C07524 ↗ChEBI CHEBI:6931 ↗ChEMBL CHEMBL655 ↗KEGG D00550 ↗DrugBank DB00683 ↗ChemSpider ↗ChEBI/ChEMBL ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗NIH ↗NIH ↗CAS 59467-64-0 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Midazolam ↗
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.