Phenazepam
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2 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA-A receptor; alpha-1/beta-2/gamma-2 | — | Ki 0.05 nM | CHEMBL | TargetGABA-A receptor; alpha-1/beta-2/gamma-2 Action— AffinityKi 0.05 nM SourceCHEMBL |
| GABA A receptor alpha-2/beta-2/gamma-2 | — | Ki 0.06 nM | CHEMBL | TargetGABA A receptor alpha-2/beta-2/gamma-2 Action— AffinityKi 0.06 nM SourceCHEMBL |
| GABA A receptor alpha-3/beta-2/gamma-2 | — | Ki 0.12 nM | CHEMBL | TargetGABA A receptor alpha-3/beta-2/gamma-2 Action— AffinityKi 0.12 nM SourceCHEMBL |
| Gamma-aminobutyric acid receptor subunit alpha-5/beta-2/gamma-2 | — | Ki 0.68 nM | CHEMBL | TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-2/gamma-2 Action— AffinityKi 0.68 nM SourceCHEMBL |
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