Baclofen
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4 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| GABA-B receptor (GABBR2) | Agonist | 7.46 IC50 | DRUGCENTRAL | TargetGABA-B receptor (GABBR2) ActionAgonist Affinity7.46 IC50 SourceDRUGCENTRAL |
| Adenosine receptor A3 (ADORA3) | — | 7.3 IC50 | DRUGCENTRAL | TargetAdenosine receptor A3 (ADORA3) Action— Affinity7.3 IC50 SourceDRUGCENTRAL |
| GABA B receptor (Gabbr2) | — | 7.52 IC50 | DRUGCENTRAL | TargetGABA B receptor (Gabbr2) Action— Affinity7.52 IC50 SourceDRUGCENTRAL |
| GABA-A receptor; anion channel (Gabrp) | — | 7.52 IC50 | DRUGCENTRAL | TargetGABA-A receptor; anion channel (Gabrp) Action— Affinity7.52 IC50 SourceDRUGCENTRAL |
External links
PubChem 2284 ↗CAS 1134-47-0 ↗ChEBI CHEBI:2972 ↗ChEMBL CHEMBL701 ↗KEGG D00241 ↗DrugBank DB00181 ↗NIH ↗NIH ↗NIH ↗ChemSpider ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗NIH ↗NIH ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗CAS 2032-34-0 ↗CAS 62594-36-9 ↗CAS 66514-99-6 ↗CAS 69308-37-8 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Baclofen ↗
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.