Buprenorphine
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| Delta-type opioid receptor (OPRD1) | Antagonist | 8.07 Ki | DRUGCENTRAL | TargetDelta-type opioid receptor (OPRD1) ActionAntagonist Affinity8.07 Ki SourceDRUGCENTRAL |
| Kappa-type opioid receptor (OPRK1) | Antagonist | 9.01 Ki | DRUGCENTRAL | TargetKappa-type opioid receptor (OPRK1) ActionAntagonist Affinity9.01 Ki SourceDRUGCENTRAL |
| Mu-type opioid receptor (OPRM1) | Partial agonist | 8.29 Ki | DRUGCENTRAL | TargetMu-type opioid receptor (OPRM1) ActionPartial agonist Affinity8.29 Ki SourceDRUGCENTRAL |
| Delta-type opioid receptor (Oprd1) | — | 9.32 Ki | DRUGCENTRAL | TargetDelta-type opioid receptor (Oprd1) Action— Affinity9.32 Ki SourceDRUGCENTRAL |
| Kappa-type opioid receptor (OPRK1) | — | 9.3 Ki | DRUGCENTRAL | TargetKappa-type opioid receptor (OPRK1) Action— Affinity9.3 Ki SourceDRUGCENTRAL |
| Mu-type opioid receptor (Oprm1) | — | 9.89 Ki | DRUGCENTRAL | TargetMu-type opioid receptor (Oprm1) Action— Affinity9.89 Ki SourceDRUGCENTRAL |
| Nociceptin receptor (OPRL1) | — | 7.11 Ki | DRUGCENTRAL | TargetNociceptin receptor (OPRL1) Action— Affinity7.11 Ki SourceDRUGCENTRAL |
| Potassium voltage-gated channel subfamily H member 2 (KCNH2) | — | 5.1 IC50 | DRUGCENTRAL | TargetPotassium voltage-gated channel subfamily H member 2 (KCNH2) Action— Affinity5.1 IC50 SourceDRUGCENTRAL |
External links
Source: DrugCentral — Buprenorphine ↗
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