DALT
Discover related
3 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| 5-hydroxytryptamine receptor 2B | — | Ki 61.66 nM | CHEMBL | Target5-hydroxytryptamine receptor 2B Action— AffinityKi 61.66 nM SourceCHEMBL |
| Sigma non-opioid intracellular receptor 1 | — | Ki 100 nM | CHEMBL | TargetSigma non-opioid intracellular receptor 1 Action— AffinityKi 100 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 1A | — | Ki 100 nM | CHEMBL | Target5-hydroxytryptamine receptor 1A Action— AffinityKi 100 nM SourceCHEMBL |
| Alpha-2A adrenergic receptor | — | Ki 123.03 nM | CHEMBL | TargetAlpha-2A adrenergic receptor Action— AffinityKi 123.03 nM SourceCHEMBL |
| Histamine H1 receptor | — | Ki 125.89 nM | CHEMBL | TargetHistamine H1 receptor Action— AffinityKi 125.89 nM SourceCHEMBL |
| Sodium-dependent serotonin transporter | — | Ki 151.36 nM | CHEMBL | TargetSodium-dependent serotonin transporter Action— AffinityKi 151.36 nM SourceCHEMBL |
| Alpha-2B adrenergic receptor | — | Ki 302 nM | CHEMBL | TargetAlpha-2B adrenergic receptor Action— AffinityKi 302 nM SourceCHEMBL |
| Unchecked | — | Ki 354.81 nM | CHEMBL | TargetUnchecked Action— AffinityKi 354.81 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 1E | — | Ki 380.19 nM | CHEMBL | Target5-hydroxytryptamine receptor 1E Action— AffinityKi 380.19 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 2C | — | Ki 389.05 nM | CHEMBL | Target5-hydroxytryptamine receptor 2C Action— AffinityKi 389.05 nM SourceCHEMBL |
| D(3) dopamine receptor | — | Ki 676.08 nM | CHEMBL | TargetD(3) dopamine receptor Action— AffinityKi 676.08 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 1D | — | Ki 691.83 nM | CHEMBL | Target5-hydroxytryptamine receptor 1D Action— AffinityKi 691.83 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 2A | — | Ki 707.95 nM | CHEMBL | Target5-hydroxytryptamine receptor 2A Action— AffinityKi 707.95 nM SourceCHEMBL |
| Alpha-2C adrenergic receptor | — | Ki 891.25 nM | CHEMBL | TargetAlpha-2C adrenergic receptor Action— AffinityKi 891.25 nM SourceCHEMBL |
| Sodium-dependent noradrenaline transporter | — | Ki 1000 nM | CHEMBL | TargetSodium-dependent noradrenaline transporter Action— AffinityKi 1000 nM SourceCHEMBL |
| Sodium-dependent dopamine transporter | — | Ki 1258.93 nM | CHEMBL | TargetSodium-dependent dopamine transporter Action— AffinityKi 1258.93 nM SourceCHEMBL |
| Alpha-1B adrenergic receptor | — | Ki 1258.93 nM | CHEMBL | TargetAlpha-1B adrenergic receptor Action— AffinityKi 1258.93 nM SourceCHEMBL |
| Alpha-1A adrenergic receptor | — | Ki 1659.59 nM | CHEMBL | TargetAlpha-1A adrenergic receptor Action— AffinityKi 1659.59 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 6 | — | Ki 1737.8 nM | CHEMBL | Target5-hydroxytryptamine receptor 6 Action— AffinityKi 1737.8 nM SourceCHEMBL |
| Kappa-type opioid receptor | — | Ki 2454.71 nM | CHEMBL | TargetKappa-type opioid receptor Action— AffinityKi 2454.71 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 7 | — | Ki 10000 nM | CHEMBL | Target5-hydroxytryptamine receptor 7 Action— AffinityKi 10000 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 5A | — | Ki 10000 nM | CHEMBL | Target5-hydroxytryptamine receptor 5A Action— AffinityKi 10000 nM SourceCHEMBL |
| Alpha-1D adrenergic receptor | — | Ki 10000 nM | CHEMBL | TargetAlpha-1D adrenergic receptor Action— AffinityKi 10000 nM SourceCHEMBL |
| 5-hydroxytryptamine receptor 1B | — | Ki 10000 nM | CHEMBL | Target5-hydroxytryptamine receptor 1B Action— AffinityKi 10000 nM SourceCHEMBL |
| Mu-type opioid receptor | — | Ki 10000 nM | CHEMBL | TargetMu-type opioid receptor Action— AffinityKi 10000 nM SourceCHEMBL |
| Histamine H3 receptor | — | Ki 10000 nM | CHEMBL | TargetHistamine H3 receptor Action— AffinityKi 10000 nM SourceCHEMBL |
| D(2) dopamine receptor | — | Ki 10000 nM | CHEMBL | TargetD(2) dopamine receptor Action— AffinityKi 10000 nM SourceCHEMBL |
Fact-sheets from PsychonautWiki. Harm-reduction reference only — not medical advice.