Pregabalin
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| Voltage-dependent calcium channel subunit alpha-2/delta-1 (CACNA2D1) | Modulator | 7.097 IC50 | DRUGCENTRAL | TargetVoltage-dependent calcium channel subunit alpha-2/delta-1 (CACNA2D1) ActionModulator Affinity7.097 IC50 SourceDRUGCENTRAL |
| Voltage-dependent calcium channel subunit alpha-2/delta-2 (CACNA2D2) | Modulator | 7.26 IC50 | DRUGCENTRAL | TargetVoltage-dependent calcium channel subunit alpha-2/delta-2 (CACNA2D2) ActionModulator Affinity7.26 IC50 SourceDRUGCENTRAL |
| Large neutral amino acids transporter small subunit 1 (SLC7A5) | — | 3.801 IC50 | DRUGCENTRAL | TargetLarge neutral amino acids transporter small subunit 1 (SLC7A5) Action— Affinity3.801 IC50 SourceDRUGCENTRAL |
| Uncharacterized protein; Voltage-dependent calcium channel alpha-2 delta subunit (CACNA2D1) | — | 7.14 IC50 | DRUGCENTRAL | TargetUncharacterized protein; Voltage-dependent calcium channel alpha-2 delta subunit (CACNA2D1) Action— Affinity7.14 IC50 SourceDRUGCENTRAL |
External links
PubChem 5486971 ↗CAS 148553-50-8 ↗ChEBI CHEBI:64356 ↗ChEMBL CHEMBL1059 ↗KEGG D02716 ↗DrugBank DB00230 ↗ChemSpider ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗NIH ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗CAS 103011-96-7 ↗CAS 128013-69-4 ↗CAS 130912-52-6 ↗CAS 1414928-41-8 ↗CAS 148553-51-9 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Pregabalin ↗
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