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Progesterone

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🧬 Receptor activity

TargetActionAffinitySource
Cation channel sperm-associated protein 1 (CATSPER1)Activator8.11 EC50DRUGCENTRAL
Cation channel sperm-associated protein 2 (CATSPER2)Activator8.11 EC50DRUGCENTRAL
Cation channel sperm-associated protein 3 (CATSPER3)Activator8.11 EC50DRUGCENTRAL
Cation channel sperm-associated protein 4 (CATSPER4)Activator8.11 EC50DRUGCENTRAL
Progesterone receptor (PGR)Agonist9.876 ED50DRUGCENTRAL
Short transient receptor potential channel 5 (TRPC5)Blocker5.3 IC50DRUGCENTRAL
Androgen receptor (AR)8.07 KiDRUGCENTRAL
C-8 sterol isomerase (ERG2)5.35 KiDRUGCENTRAL
Corticosteroid-binding globulin (SERPINA6)7.38 KiDRUGCENTRAL
Estrogen receptor (ESR1)DRUGCENTRAL
Fatty acid-binding protein, intestinal (FABP2)4.7 KiDRUGCENTRAL
Fatty acid-binding protein, liver (Fabp1)7.57 KiDRUGCENTRAL
Glucocorticoid receptor (NR3C1)7.52 KiDRUGCENTRAL
Mineralocorticoid receptor (NR3C2)11 EC50DRUGCENTRAL
Multidrug resistance protein 1 (ABCB1)4.32 IC50DRUGCENTRAL
P2X purinoceptor 3 (P2RX3)5.8 IC50DRUGCENTRAL
Progesterone receptor (PGR)8.441 KiDRUGCENTRAL
Sex hormone-binding globulin (SHBG)6.94 KdDRUGCENTRAL
Sigma non-opioid intracellular receptor 1 (SIGMAR1)6.59 KiDRUGCENTRAL
Sodium/nucleoside cotransporter 1 (SLC28A1)5.174 KiDRUGCENTRAL
Steroid 5-alpha-reductase (Srd5a1)5.8 IC50DRUGCENTRAL
Sterol O-acyltransferase 1 (SOAT1)4.77 IC50DRUGCENTRAL
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Source: DrugCentral — Progesterone ↗

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