Melatonin
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5 sources
🧬 Receptor activity
| Target | Action | Affinity | Source | |
|---|---|---|---|---|
| 5-hydroxytryptamine receptor 2B (HTR2B) | Antagonist | 5.2 Ki | DRUGCENTRAL | Target5-hydroxytryptamine receptor 2B (HTR2B) ActionAntagonist Affinity5.2 Ki SourceDRUGCENTRAL |
| Melatonin receptor type 1A (MTNR1A) | Agonist | 9.4 EC50 | DRUGCENTRAL | TargetMelatonin receptor type 1A (MTNR1A) ActionAgonist Affinity9.4 EC50 SourceDRUGCENTRAL |
| Melatonin receptor type 1B (MTNR1B) | Agonist | 9.7 EC50 | DRUGCENTRAL | TargetMelatonin receptor type 1B (MTNR1B) ActionAgonist Affinity9.7 EC50 SourceDRUGCENTRAL |
| Cytochrome P450 1B1 (CYP1B1) | — | 4.85 Ki | DRUGCENTRAL | TargetCytochrome P450 1B1 (CYP1B1) Action— Affinity4.85 Ki SourceDRUGCENTRAL |
| Histamine H3 receptor (HRH3) | — | 9.3 Ki | DRUGCENTRAL | TargetHistamine H3 receptor (HRH3) Action— Affinity9.3 Ki SourceDRUGCENTRAL |
| Melatonin receptor | — | 9.75 Ki | DRUGCENTRAL | TargetMelatonin receptor Action— Affinity9.75 Ki SourceDRUGCENTRAL |
| Melatonin receptor type 1B | — | 9.15 Ki | DRUGCENTRAL | TargetMelatonin receptor type 1B Action— Affinity9.15 Ki SourceDRUGCENTRAL |
| Myeloperoxidase (MPO) | — | 5.52 IC50 | DRUGCENTRAL | TargetMyeloperoxidase (MPO) Action— Affinity5.52 IC50 SourceDRUGCENTRAL |
| Nuclear receptor ROR-alpha (RORA) | — | 9 EC50 | DRUGCENTRAL | TargetNuclear receptor ROR-alpha (RORA) Action— Affinity9 EC50 SourceDRUGCENTRAL |
| Ribosyldihydronicotinamide dehydrogenase [quinone] (NQO2) | — | 7.56 Ki | DRUGCENTRAL | TargetRibosyldihydronicotinamide dehydrogenase [quinone] (NQO2) Action— Affinity7.56 Ki SourceDRUGCENTRAL |
External links
PubChem 896 ↗CAS 73-31-4 ↗CAS 8041-44-9 ↗KEGG C01598 ↗ChEBI CHEBI:16796 ↗ChEMBL CHEMBL45 ↗KEGG D08170 ↗DrugBank DB01065 ↗NIH ↗NIH ↗NIH ↗NIH ↗ChemSpider ↗ChEBI/ChEMBL ↗ChEBI/ChEMBL ↗Guide to Pharmacology ↗Guide to Pharmacology ↗NIH ↗NIH ↗NIH ↗NIH ↗DrugBank ↗ChEBI/ChEMBL ↗NIH ↗NIH ↗NIH ↗NIH ↗NIH ↗NIH ↗NIH ↗NIH ↗NIH ↗CAS 51023-76-8 ↗CAS 66521-38-8 ↗PsychonautWiki ↗Erowid ↗Experience reports (PiHKAL) ↗Experience reports (TiHKAL) ↗
Source: DrugCentral — Melatonin ↗
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